Patents
274 patents filed by Insilico Medicine and related entities, of which 58 list Alex Zhavoronkov as a named inventor.
| Pub. Number | Title | Assignee | Date | Role |
|---|---|---|---|---|
| n/a | KINASE INHIBITORS | n/a | n/a | Inventor |
| n/a | METHOD AND MEDICAMENT FOR TREATING ENDOMETRIOSIS | n/a | n/a | Inventor |
| n/a | METHOD AND MEDICAMENT FOR TREATING ENDOMETRIOSIS | n/a | n/a | Inventor |
| n/a | METHOD AND MEDICAMENT FOR TREATING ENDOMETRIOSIS | n/a | n/a | Inventor |
| n/a | METHODS AND SYSTEMS FOR ALCHEMICAL BINDING FREE ENERGY | n/a | n/a | Inventor |
| n/a | Subset conditioning using variational autoencoder with a learnable tensor train induced prior | n/a | n/a | Inventor |
| n/a | Methods of inhibiting kinases | n/a | n/a | Inventor |
| n/a | Subset conditioning using variational autoencoder with a learnable tensor train induced prior | n/a | n/a | Inventor |
| n/a | Kinase inhibitors | n/a | n/a | Inventor |
| n/a | LOCAL STEPS IN LATENT SPACE AND DESCRIPTORS-BASED MOLECULES FILTERING FOR CONDITIONAL MOLECULAR GENERATION | n/a | n/a | Inventor |
| n/a | Analogs for the treatment of disease | n/a | n/a | Inventor |
| n/a | Analogs for the treatment of disease | n/a | n/a | Inventor |
| n/a | Mutual information adversarial autoencoder | n/a | n/a | Inventor |
| n/a | Analogs for the treatment of disease | n/a | n/a | Inventor |
| n/a | ANALOGS FOR THE TREATMENT OF DISEASE | n/a | n/a | Inventor |
| n/a | ANALOGS FOR THE TREATMENT OF DISEASE | n/a | n/a | Inventor |
| n/a | ANALOGS FOR THE TREATMENT OF DISEASE | n/a | n/a | Inventor |
| n/a | ANALOGS FOR THE TREATMENT OF DISEASE | n/a | n/a | Inventor |
| n/a | ADVERSARIAL FRAMEWORK FOR MOLECULAR CONFORMATION SPACE MODELING IN INTERNAL COORDINATES | n/a | n/a | Inventor |
| n/a | ANALOGS FOR THE TREATMENT OF DISEASE | n/a | n/a | Inventor |
| n/a | METHOD AND MEDICAMENT FOR TREATING AMYOTROPHIC LATERAL SCLEROSIS | n/a | n/a | Inventor |
| n/a | TLR 9 inhibitors | n/a | n/a | Inventor |
| n/a | Bycyclic JAK inhibitors and uses thereof | n/a | n/a | Inventor |
| n/a | EDGE MESSAGE PASSING NEURAL NETWORK | n/a | n/a | Inventor |
| n/a | SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS | n/a | n/a | Inventor |
| n/a | RETROSYNTHESIS-RELATED SYNTHETIC ACCESSIBILITY | n/a | n/a | Inventor |
| n/a | SCAFFOLD-ORIENTED UNIVERSAL LINE SYSTEM | n/a | n/a | Inventor |
| n/a | ADVERSARIAL AUTOENCODER ARCHITECTURE FOR METHODS OF GRAPH TO SEQUENCE MODELS | n/a | n/a | Inventor |
| n/a | DETERMINISTIC DECODER VARIATIONAL AUTOENCODER | n/a | n/a | Inventor |
| n/a | EDGE MESSAGE PASSING NEURAL NETWORK | n/a | n/a | Inventor |
| n/a | SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS | n/a | n/a | Inventor |
| n/a | BIOLOGICAL DATA SIGNATURES OF AGING AND METHODS OF DETERMINING A BIOLOGICAL AGING CLOCK | n/a | n/a | Inventor |
| n/a | TLR inhibitors | n/a | n/a | Inventor |
| n/a | TLR 9 inhibitors | n/a | n/a | Inventor |
| n/a | Methods of inhibiting kinases | n/a | n/a | Inventor |
| n/a | KINASE INHIBITORS | n/a | n/a | Inventor |
| n/a | KINASE INHIBITORS | n/a | n/a | Inventor |
| n/a | SYNTHETIC BIOLOGICAL CHARACTERISTIC GENERATOR BASED ON REAL BIOLOGICAL DATA SIGNATURES | n/a | n/a | Inventor |
| n/a | WORKFLOW FOR GENERATING COMPOUNDS WITH BIOLOGICAL ACTIVITY AGAINST A SPECIFIC BIOLOGICAL TARGET | n/a | n/a | Inventor |
| n/a | WORKFLOW FOR GENERATING COMPOUNDS WITH BIOLOGICAL ACTIVITY AGAINST A SPECIFIC BIOLOGICAL TARGET | n/a | n/a | Inventor |
| n/a | TLR INHIBITORS | n/a | n/a | Inventor |
| n/a | KINASE INHIBITORS | n/a | n/a | Inventor |
| n/a | METHODS OF INHIBITING KINASES | n/a | n/a | Inventor |
| n/a | BICYCLIC JAK INHIBITORS AND USES THEREOF | n/a | n/a | Inventor |
| n/a | WORKFLOW FOR GENERATING COMPOUNDS WITH BIOLOGICAL ACTIVITY AGAINST A SPECIFIC BIOLOGICAL TARGET | n/a | n/a | Inventor |
| n/a | Deep proteome markers of human biological aging and methods of determining a biological aging clock | n/a | n/a | Inventor |
| n/a | TLR inhibitors | n/a | n/a | Inventor |
| n/a | MUTUAL INFORMATION ADVERSARIAL AUTOENCODER | n/a | n/a | Inventor |
| n/a | SUBSET CONDITIONING USING VARIATIONAL AUTOENCODER WITH A LEARNABLE TENSOR TRAIN INDUCED PRIOR | n/a | n/a | Inventor |
| n/a | Deep transcriptomic markers of human biological aging and methods of determining a biological aging clock | n/a | n/a | Inventor |
| n/a | Method of treating senescence with multi-stage longevity therapeutics | n/a | n/a | Inventor |
| n/a | Mutual information adversarial autoencoder | n/a | n/a | Inventor |
| n/a | SYSTEM, METHOD AND SOFTWARE FOR ANALYSIS OF INTRACELLULAR SIGNALING PATHWAY ACTIVATION USING TRANSCRIPTOMIC DATA | n/a | n/a | Inventor |
| n/a | SYSTEMS, METHODS AND SOFTWARE FOR RANKING POTENTIAL GEROPROTECTIVE DRUGS | n/a | n/a | Inventor |
| n/a | SYSTEM, METHOD AND SOFTWARE FOR ANALYSIS OF INTRACELLULAR SIGNALING PATHWAY ACTIVATION USING TRANSCRIPTOMIC DATA | n/a | n/a | Inventor |
| n/a | SYSTEM, METHOD AND SOFTWARE FOR ANALYSIS OF INTRACELLULAR SIGNALING PATHWAY ACTIVATION USING TRANSCRIPTOMIC DATA | n/a | n/a | Inventor |
| n/a | SYSTEM, METHOD AND SOFTWARE FOR PREDICTING DRUG EFFICACY IN A PATIENT | n/a | n/a | Inventor |
| n/a | Systems and methods for communicating with a computer using brain activity patterns | n/a | n/a | Inventor |
| n/a | NOVEL COMPOUNDS AS GLUCOCORTICOID RECEPTOR MODULATORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE CYCLIN-DEPENDENT KINASE (CDK) 12 AND/OR CDK13 INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CYCLIN-DEPENDENT KINASE (CDK) 12 AND/OR CDK13 INHIBITOR COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | TEAD INHIBITOR COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | TEAD INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE TEAD INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS CYCLIC GMP-AMP SYNTHASE INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | WERNER SYNDROME RECQ HELICASE (WRN) INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | SCALABLE FRAMEWORK FOR 3D MOLECULAR DESIGN VIA LANGUAGE MODELING AND REINFORCEMENT LEARNING | n/a | n/a | Assignee |
| n/a | HETEROCYCLIC INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) IN COMBINATION WITH ADDITIONAL AGENTS FOR USE IN THE TREATMENT OF… | n/a | n/a | Assignee |
| n/a | NLRP3 INFLAMMASOME INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SALT-INDUCIBLE KINASES (SIK) INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | SALT-INDUCIBLE KINASES (SIK) INHIBITORS | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS SALT-INDUCIBLE KINASES INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | WERNER SYNDROME RECQ HELICASE (WRN) INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS KRAS INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF KIF18A AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRBN-BINDING COMPOUNDS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS GLP-1R AGONISTS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS NLRP3 INFLAMMASOME INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | TNIK INHIBITORS FOR THE TREATMENT OF PAIN | n/a | n/a | Assignee |
| n/a | ADVANCED RETROSYNTHESIS-RELATED SYNTHETIC ACCESSIBILITY MODELING | n/a | n/a | Assignee |
| n/a | PHARMACEUTICAL COMBINATIONS FOR USE IN THE TREATMENT OF CANCERS | n/a | n/a | Assignee |
| n/a | GLUCOSE-DEPENDENT INSULINOTROPIC POLYPEPTIDE RECEPTOR (GIPR) ANTAGONISTS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF KIF18A AND USES THEREOF | n/a | n/a | Assignee |
| n/a | NLRP3 INFLAMMASOME INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF FGFR2 AND FGFR3 AND USES THEREOF | n/a | n/a | Assignee |
| n/a | LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITOR, COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITOR COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS, COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SPIRO DERIVATIVES AS WRN INHIBITORS | n/a | n/a | Assignee |
| n/a | NLRP3 INFLAMMASOME INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PRMT5 INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF KIF18A AND USES THEREOF | n/a | n/a | Assignee |
| n/a | MPRO INHIBITORS FOR TREATING CORONAVIRUS INFECTIONS | n/a | n/a | Assignee |
| n/a | CDK8/19 DUAL INHIBITORS AND METHODS OF USE THEREOF | n/a | n/a | Assignee |
| n/a | NLRP3 INFLAMMASOME INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF FGFR2 AND FGFR3 AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE METHIONINE ADENOSYLTRANSFERASE 2a (MAT2A) INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITOR COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITOR, COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE SARS-COV-2 INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS, COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS, COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SPIRO DERIVATIVES AS WRN INHIBITORS | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | NLRP3 INFLAMMASOME INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PRMT5 INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | KRAS INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SYNTHESIS OF MACROCYCLIC COMPOUND AND MEDICAL USE OF MACROCYCLIC COMPOUND | n/a | n/a | Assignee |
| n/a | SUBSTITUTED THIAZOLE COMPOUNDS AS CDK2/4/6 INHIBITORS AND METHODS OF USE THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE TNIK INHIBITOR AND USES THEREOF | n/a | n/a | Assignee |
| n/a | ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PHARMACEUTICAL FORMULATIONS FOR INHALATION AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYSTALLINE BETA-LACTAM DERIVATIVES AND USES THEREOF | n/a | n/a | Assignee |
| n/a | ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CRYTSALLINE FORMS OF ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | FUSED RING COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF | n/a | n/a | Assignee |
| n/a | BIFUNCTIONAL COMPOUNDS FOR TARGETING PKMYT1 AND METHODS OF USE | n/a | n/a | Assignee |
| n/a | COMBINATIONS TREATMENTS OF DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND OTHER THERAPIES | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS PKMYT1 INHIBITORS AND USE THEREOF | n/a | n/a | Assignee |
| n/a | 3CL-PROTEASE INHIBITORS FOR TREATING OR PREVENTING VETERINARY CORONAVIRUS INFECTIONS | n/a | n/a | Assignee |
| n/a | CBL-B INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS MODULATORS OF SODIUM CHANNELS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS GLP-1R AGONISTS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | NOVEL COMPOUNDS AS GLP-1R AGONISTS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SARS-CoV-2 inhibitors for treating coronavirus infections | n/a | n/a | Assignee |
| n/a | Prolyl hydroxylase domain-containing protein (PHD) inhibitors and uses thereof | n/a | n/a | Assignee |
| n/a | Small molecule inhibitors of ubiquitin specific protease 1 (USP1) and uses thereof | n/a | n/a | Assignee |
| n/a | Prolyl hydroxylase domain-containing protein (PHD) inhibitors and uses thereof | n/a | n/a | Assignee |
| n/a | Beta-lactam derivatives for the treatment of diseases | n/a | n/a | Assignee |
| n/a | Methionine adenosyltransferase 2a (MAT2A) inhibitors and uses thereof | n/a | n/a | Assignee |
| n/a | Prolyl hydroxylase domain-containing protein (PHD) inhibitors and uses thereof | n/a | n/a | Assignee |
| n/a | Diacylglycerol kinase (DGK) alpha inhibitors and uses thereof | n/a | n/a | Assignee |
| n/a | Lysine acetyltransferase 6A (KAT6A) inhibitors and uses thereof | n/a | n/a | Assignee |
| n/a | TEAD inhibitors and methods of uses thereof | n/a | n/a | Assignee |
| n/a | Beta-lactam derivatives for the treatment of diseases | n/a | n/a | Assignee |
| n/a | Structure-based deep generative model for binding site descriptors extraction and de novo molecular generation | n/a | n/a | Assignee |
| n/a | Small molecule inhibitors of ubiquitin specific protease 1 (USP1) and uses thereof | n/a | n/a | Assignee |
| n/a | ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | MEMBRANE-ASSOCIATED TYROSINE-AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | MEMBRANE-ASSOCIATED TYROSINE-AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PYRAZOLE MEMBRANE-ASSOCIATED TYROSINE-AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PYRAZOLE MEMBRANE-ASSOCIATED TYROSINE-AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF FGFR2 AND FGFR3 AND USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF CYCLIN-DEPENDENT KINASE (CDK) 12 AND/OR CDK13 AND USES THEREOF | n/a | n/a | Assignee |
| n/a | METHODS OF MANUFACTURING KINASE INHIBITORS | n/a | n/a | Assignee |
| n/a | SALT-INDUCIBLE KINASES (SIK) INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | SPIRO DERIVATIVE AS KIF18A INHIBITOR | n/a | n/a | Assignee |
| n/a | INHIBITORS OF KIF18A AND USES THEREOF | n/a | n/a | Assignee |
| n/a | ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | MEMBRANE-ASSOCIATED TYROSINE-AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | STRUCTURE-BASED DEEP GENERATIVE MODEL FOR BINDING SITE DESCRIPTORS EXTRACTION AND DE NOVO MOLECULAR GENERATION | n/a | n/a | Assignee |
| n/a | DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | HETEROAROMATIC COMPOUNDS AS PKMYT1 INHIBITORS AND USE THEREOF | n/a | n/a | Assignee |
| n/a | PYRAZOLE MEMBRANE-ASSOCIATED TYROSINE-AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | HPK1 ANTAGONISTS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CDK8/19 DUAL INHIBITORS AND METHODS OF USE THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF FGFR2 AND FGFR3 AND USES THEREOF | n/a | n/a | Assignee |
| n/a | CBL-B INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF CYCLIN-DEPENDENT KINASE (CDK) 12 AND/OR CDK13 AND USES THEREOF | n/a | n/a | Assignee |
| n/a | METHODS OF MANUFACTURING KINASE INHIBITORS | n/a | n/a | Assignee |
| n/a | INHIBITORS OF TREX1 AND USES THEREOF | n/a | n/a | Assignee |
| n/a | TEAD INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE 1 (ENPP1) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | NLRP3 INFLAMMASOME INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SALT-INDUCIBLE KINASES (SIK) INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | SPIRO DERIVATIVE AS KIF18A INHIBITOR | n/a | n/a | Assignee |
| n/a | CBL-B INHIBITORS AND METHODS OF USES THEREOF | n/a | n/a | Assignee |
| n/a | SPIROCYCLIC HPK1 ANTAGONISTS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | INHIBITORS OF KIF18A AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | BETA-LACTAM DERIVATIVES FOR THE TREATMENT OF DISEASES | n/a | n/a | Assignee |
| n/a | BETA-LACTAM DERIVATIVES FOR THE TREATMENT OF DISEASES | n/a | n/a | Assignee |
| n/a | METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SARS-COV-2 INHIBITORS FOR TREATING CORONAVIRUS INFECTIONS | n/a | n/a | Assignee |
| n/a | SARS-COV-2 INHIBITORS FOR TREATING CORONAVIRUS INFECTIONS | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE | n/a | n/a | Assignee |
| n/a | PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE | n/a | n/a | Assignee |
| n/a | ANALOGS FOR THE TREATMENT OF DISEASE | n/a | n/a | Assignee |
| n/a | ADVERSARIAL FRAMEWORK FOR MOLECULAR CONFORMATION SPACE MODELING IN INTERNAL COORDINATES | n/a | n/a | Assignee |
| n/a | BETA-LACTAM DERIVATIVES FOR THE TREATMENT OF DISEASES | n/a | n/a | Assignee |
| n/a | METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | PROLYL HYDROXYLASE DOMAIN-CONTAINING PROTEIN (PHD) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SARS-COV-2 INHIBITORS FOR TREATING CORONAVIRUS INFECTIONS | n/a | n/a | Assignee |
| n/a | SARS-COV-2 INHIBITORS FOR TREATING CORONAVIRUS INFECTIONS | n/a | n/a | Assignee |
| n/a | CDK8/19 DUAL INHIBITORS AND METHODS OF USE | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SMALL MOLECULE INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 1 (USP1) AND USES THEREOF | n/a | n/a | Assignee |
| n/a | LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | SUBSTITUTED MONOCYCLIC OR BICYCLIC HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF | n/a | n/a | Assignee |
| n/a | Retrosynthesis systems and methods | n/a | n/a | Assignee |
| n/a | SCAFFOLD-ORIENTED UNIVERSAL LINE SYSTEM | n/a | n/a | Assignee |
| n/a | ADVERSARIAL AUTOENCODER ARCHITECTURE FOR METHODS OF GRAPH TO SEQUENCE MODELS | n/a | n/a | Assignee |
| n/a | DETERMINISTIC DECODER VARIATIONAL AUTOENCODER | n/a | n/a | Assignee |
| n/a | SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS | n/a | n/a | Assignee |
| n/a | GRAPH NORMALIZING FLOW FOR HIERARCHICAL MOLECULAR GENERATION | n/a | n/a | Assignee |
| n/a | RETROSYNTHESIS SYSTEMS AND METHODS | n/a | n/a | Assignee |
| n/a | RETROSYNTHESIS-RELATED SYNTHETIC ACCESSIBILITY | n/a | n/a | Assignee |
| n/a | TLR 9 INHIBITORS | n/a | n/a | Assignee |
| n/a | GRAPH NORMALIZING FLOW FOR HIERARCHICAL MOLECULAR GENERATION | n/a | n/a | Assignee |
| n/a | METHYLATION DATA SIGNATURES OF AGING AND METHODS OF DETERMINING A METHYLATION AGING CLOCK | n/a | n/a | Assignee |
| n/a | RETROSYNTHESIS SYSTEMS AND METHODS | n/a | n/a | Assignee |
| n/a | Kinase inhibitors | n/a | n/a | Assignee |
| n/a | Scaffold-oriented universal line system | n/a | n/a | Assignee |
| n/a | Workflow for generating compounds with biological activity against a specific biological target | n/a | n/a | Assignee |
| n/a | TLR INHIBITORS | n/a | n/a | Assignee |
| n/a | TLR INHIBITORS | n/a | n/a | Assignee |
| n/a | BICYCLIC JAK INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | BICYCLIC JAK INHIBITORS AND USES THEREOF | n/a | n/a | Assignee |
| n/a | DEEP PROTEOME MARKERS OF HUMAN BIOLOGICAL AGING AND METHODS OF DETERMINING A BIOLOGICAL AGING CLOCK | n/a | n/a | Assignee |
| n/a | DEEP PROTEOME MARKERS OF HUMAN BIOLOGICAL AGING AND METHODS OF DETERMINING A BIOLOGICAL AGING CLOCK | n/a | n/a | Assignee |
| n/a | SYNTHETIC BIOLOGICAL CHARACTERISTIC GENERATOR BASED ON REAL BIOLOGICAL DATA SIGNATURES | n/a | n/a | Assignee |
| n/a | DEEP PROTEOME MARKERS OF HUMAN BIOLOGICAL AGING AND METHODS OF DETERMINING A BIOLOGICAL AGING CLOCK | n/a | n/a | Assignee |
| n/a | SYNTHETIC BIOLOGICAL CHARACTERISTIC GENERATOR BASED ON REAL BIOLOGICAL DATA SIGNATURES | n/a | n/a | Assignee |
| n/a | KINASE INHIBITORS AND METHODS OF SYNTHESIS AND TREATMENT | n/a | n/a | Assignee |
| n/a | Kinase inhibitors | n/a | n/a | Assignee |
| n/a | Entangled conditional adversarial autoencoder for drug discovery | n/a | n/a | Assignee |
| n/a | MUTUAL INFORMATION ADVERSARIAL AUTOENCODER | n/a | n/a | Assignee |
| n/a | MUTUAL INFORMATION ADVERSARIAL AUTOENCODER | n/a | n/a | Assignee |
| n/a | SUBSET CONDITIONING USING VARIATIONAL AUTOENCODER WITH A LEARNABLE TENSOR TRAIN INDUCED PRIOR | n/a | n/a | Assignee |
| n/a | SUBSET CONDITIONING USING VARIATIONAL AUTOENCODER WITH A LEARNABLE TENSOR TRAIN INDUCED PRIOR | n/a | n/a | Assignee |
| n/a | KINASE INHIBITORS | n/a | n/a | Assignee |
| n/a | Subset conditioning using variational autoencoder with a learnable tensor train induced prior | n/a | n/a | Assignee |
| n/a | Withaferin compositions for prevention of aging | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |
| n/a | n/a | n/a | n/a | Assignee |